SCHEMBL13460360

SCHEMBL13460360

Cc1ccc(C#N)cc1Oc1ccc2c(c1)B(O)OC2

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.58
PDE4A P27815 4/20 0.58
PDE4C Q08493 4/20 0.58
PDE4D Q08499 4/20 0.58
CHRM1 P11229 1/20 0.58
ADRA1A P35348 1/20 0.58
PDE1A P54750 1/20 0.58
PDE3B Q13370 1/20 0.58
PDE7A Q13946 1/20 0.58
PDE3A Q14432 1/20 0.58
ROCK2 O75116 2/20 0.48
ROCK1 Q13464 2/20 0.48
KLK1 P06870 1/20 0.47
KLK5 Q9Y337 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5583333 0.84 PDE4B (0.80) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL595831 0.84 PDE4B (0.80) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2229887 0.84 ROCK2 (0.65) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2230863 0.84 ROCK2 (0.65) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL8378290 0.81 PDE4B (0.72) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL594783 0.81 PDE4B (0.81) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL5134350 0.81 PDE4B (0.81) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL13111023 0.80 PDE4A (0.54) PDE4BPDE4APDE4CPDE4DROCK2
SCHEMBL1232022 0.79 PDE4B (0.58) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2532271 0.78 PDE4B (0.70) PDE4BPDE4APDE4CPDE4DCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028005-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2010-03-11 WO disclosed