SCHEMBL13460751

SCHEMBL13460751

CCCOc1ccc(C(=O)NCc2cc(-c3cccc(C=O)c3)ccc2O)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
MAPT P10636 2/20 0.41
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
ROCK2 O75116 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ROCK1 Q13464 1/20 0.38
ERN1 O75460 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NPC1 O15118 3/20 0.38
PPARG P37231 1/20 0.37
RAB9A P51151 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13461061 0.93 TP53 (0.43) TP53MAPTPPARDPPARAROCK2
SCHEMBL13460849 0.91 PPARD (0.47) TP53MAPTPPARDPPARAPPARG
SCHEMBL13460876 0.90 PPARD (0.45) TP53MAPTPPARDPPARAROCK2
SCHEMBL13460883 0.90 PPARD (0.44) TP53MAPTPPARDPPARANPC1
SCHEMBL13460848 0.87 PPARD (0.41) TP53MAPTPPARDPPARAROCK2
SCHEMBL3417430 0.86 PPARD (0.52) TP53MAPTPPARDPPARAPPARG
SCHEMBL13460801 0.86 TP53 (0.41) TP53MAPTPPARDPPARAROCK2
SCHEMBL13461056 0.84 PPARD (0.45) TP53PPARDPPARAPPARGADRB1
SCHEMBL13460949 0.84 HPGD (0.44) TP53MAPTROCK2CYP3A4CYP2D6
SCHEMBL13460940 0.83 PPARD (0.46) TP53MAPTPPARDPPARANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed