SCHEMBL13467656

SCHEMBL13467656

COc1ccc2c(Cc3ccc(NC(=O)c4c(C)n(CC(C)=O)n(-c5ccccc5)c4=O)cc3F)ccnc2c1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.79
KDR P35968 20/20 0.79
IGF1R P08069 19/20 0.70
MST1R Q04912 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13467647 0.93 MET (0.68) METKDRIGF1RMST1R
SCHEMBL13467869 0.91 MET (0.68) METKDRIGF1RMST1R
SCHEMBL13467862 0.91 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467625 0.90 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467868 0.90 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467609 0.90 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467705 0.89 MET (0.71) METKDRIGF1RMST1R
SCHEMBL198809 0.88 MET (1.00) METKDRIGF1RMST1R
SCHEMBL13467880 0.85 MET (0.67) METKDRIGF1RMST1R
SCHEMBL13467863 0.83 MET (0.61) METKDRIGF1RMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881976-B1 SUBSTITUTED AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS AMGEN INC (US) 2012-10-17 EP disclosed