SCHEMBL13467705

SCHEMBL13467705

COc1ccc2c(Cc3ccc(NC(=O)c4c(C)n(CC(C)(O)CO)n(-c5ccccc5)c4=O)cc3F)ccnc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.71
KDR P35968 19/20 0.71
IGF1R P08069 17/20 0.71
MST1R Q04912 2/20 0.71
AURKA O14965 1/20 0.58
JAK2 O60674 1/20 0.58
RPS6KA5 O75582 1/20 0.58
ABL1 P00519 1/20 0.58
INSR P06213 1/20 0.58
LCK P06239 1/20 0.58
FES P07332 1/20 0.58
CSF1R P07333 1/20 0.58
LYN P07948 1/20 0.58
RET P07949 1/20 0.58
FGR P09769 1/20 0.58
KIT P10721 1/20 0.58
PIM1 P11309 1/20 0.58
FGFR1 P11362 1/20 0.58
SRC P12931 1/20 0.58
PRKACA P17612 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13467625 0.94 MET (0.79) METKDRIGF1RMST1RAURKA
SCHEMBL13467656 0.89 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467862 0.89 MET (0.79) METKDRIGF1RMST1R
SCHEMBL199850 0.89 MET (0.90) METKDRIGF1RMST1RAXL
SCHEMBL13467868 0.88 MET (0.79) METKDRIGF1RMST1R
SCHEMBL13467647 0.88 MET (0.68) METKDRIGF1RMST1R
SCHEMBL13467609 0.87 MET (0.79) METKDRIGF1RMST1R
SCHEMBL198003 0.84 MET (0.89) METKDRIGF1RMST1RAXL
SCHEMBL199079 0.83 MET (1.00) METKDRIGF1RMST1RAURKA
SCHEMBL29383141 0.83 MET (1.00) METKDRIGF1RMST1RAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881976-B1 SUBSTITUTED AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS AMGEN INC (US) 2012-10-17 EP disclosed