SCHEMBL1349065

SCHEMBL1349065

CC(C)(CO)NS(=O)(=O)c1cncc(C#Cc2cnn3c(C4CC4)cc(-c4ccc(Cl)cc4)nc23)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.36
PSD A5PKW4 2/20 0.33
KMT2A Q03164 1/20 0.33
KIF18A Q8NI77 1/20 0.32
KDM1A O60341 2/20 0.32
MAOA P21397 2/20 0.32
PIK3CD O00329 2/20 0.31
PIK3CB P42338 2/20 0.31
PIK3CG P48736 2/20 0.31
PIK3CA P42336 1/20 0.31
CSNK2A1 P68400 1/20 0.31
ALPG P10696 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
DUT P33316 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1348942 0.94 PTGDR2 (0.36) PTGDR2PSDKDM1AMAOAPIK3CD
SCHEMBL1349423 0.92 PLAT (0.33) PTGDR2KIF18APIK3CDPIK3CBPIK3CG
SCHEMBL1346123 0.91 KIF18A (0.38) PTGDR2PSDKMT2AKIF18ADUT
SCHEMBL1349026 0.86 PLAT (0.33) PTGDR2KIF18APIK3CDPIK3CBPIK3CG
SCHEMBL1348328 0.85 PTGDR2 (0.35) PTGDR2PSDCSNK2A1
SCHEMBL2828897 0.85 PTGDR2 (0.36) PTGDR2PSDCSNK2A1
SCHEMBL1347269 0.84 PTGDR2 (0.39) PTGDR2KIF18AKDM1AMAOAPIK3CD
SCHEMBL1348244 0.84 PSD (0.32) PSDKMT2AKIF18ACSNK2A1DUT
SCHEMBL1348707 0.83 PSD (0.36) PTGDR2PSDCSNK2A1
SCHEMBL1348454 0.80 HPGD (0.41) KMT2AKIF18ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4801724-B2 2011-10-26 JP claimed
EP-1863818-B1 ACETYLENYL-PYRAZOLO-PVRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-03-10 EP claimed
US-8063048-B2 Acetylenyl-pyrazolo-pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-11-22 US disclosed