SCHEMBL1348942

SCHEMBL1348942

CC(CO)(CO)NS(=O)(=O)c1cncc(C#Cc2cnn3c(C4CC4)cc(-c4ccc(Cl)cc4)nc23)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.36
PSD A5PKW4 3/20 0.33
KDM1A O60341 2/20 0.32
MAOA P21397 2/20 0.32
PIK3CD O00329 2/20 0.31
PIK3CB P42338 2/20 0.31
PIK3CG P48736 2/20 0.31
PIK3CA P42336 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1349065 0.94 PTGDR2 (0.36) PTGDR2PSDKDM1AMAOAPIK3CD
SCHEMBL1349026 0.92 PLAT (0.33) PTGDR2PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL1349423 0.86 PLAT (0.33) PTGDR2PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL1346123 0.85 KIF18A (0.38) PTGDR2PSDCA12CA9
SCHEMBL2828897 0.85 PTGDR2 (0.36) PTGDR2PSDCSNK2A1
SCHEMBL1348707 0.83 PSD (0.36) PTGDR2PSDCSNK2A1CA12CA9
SCHEMBL1347485 0.80 HPGD (0.41)
SCHEMBL1348434 0.80 HPGD (0.38)
SCHEMBL1348328 0.79 PTGDR2 (0.35) PTGDR2PSDCSNK2A1
SCHEMBL1348311 0.79 LMNA (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4801724-B2 2011-10-26 JP claimed
EP-1863818-B1 ACETYLENYL-PYRAZOLO-PVRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-03-10 EP claimed
US-8063048-B2 Acetylenyl-pyrazolo-pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-11-22 US disclosed