SCHEMBL13509357

SCHEMBL13509357

C=C(S)NC(=O)c1cccc2oc(-c3cc(F)ccc3C(F)(F)F)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.38
TOP2A P11388 2/20 0.37
KCNH2 Q12809 2/20 0.35
CYP3A4 P08684 1/20 0.35
CREBBP Q92793 1/20 0.35
MAPT P10636 4/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGES O14684 2/20 0.34
S1PR1 P21453 1/20 0.33
RAB9A P51151 4/20 0.32
NPC1 O15118 3/20 0.32
KMT2A Q03164 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 2/20 0.32
GLA P06280 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548008 0.80 GRM5 (0.45) MAPTALDH1A1LMNAPOLBPTGES
SCHEMBL4548007 0.79 NPC1 (0.45) MAPTALDH1A1RAB9ANPC1KMT2A
SCHEMBL4548010 0.73 JAK2 (0.41) HTR3AKCNH2ALDH1A1PTGESRAB9A
SCHEMBL4548004 0.72 GRM5 (0.45) MAPTALDH1A1LMNAPOLBPTGES
SCHEMBL4548009 0.71 WDR5 (0.40) ALDH1A1RAB9ANPC1KMT2AMEN1
SCHEMBL4548003 0.71 GAA (0.47) MAPTALDH1A1RAB9ANPC1KMT2A
SCHEMBL442097 0.70 TOP2A (0.52) TOP2AALDH1A1KDM4EHPGD
SCHEMBL1937623 0.68 TOP2A (0.68) HTR3ATOP2AKCNH2CYP3A4MAPT
SCHEMBL4547998 0.68 GRM5 (0.48) TOP2AMAPTALDH1A1POLBPTGES
SCHEMBL1936924 0.66 CYP1A2 (0.50) MAPTALDH1A1POLBRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010019606-A1 BENZOXAZOLES, BENZTHIAZOLES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2010-02-18 WO disclosed