SCHEMBL13544006

SCHEMBL13544006

O=C(C1CCCC1)N1CCC(OCCN2CCC3(CC2)C(=O)NCN3c2ccccc2)(c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.92

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.92
OPRM1 P35372 4/20 0.54
OPRL1 P41146 4/20 0.54
SLC6A9 P48067 2/20 0.54
SLC6A5 Q9Y345 2/20 0.54
OPRD1 P41143 3/20 0.49
OPRK1 P41145 3/20 0.49
PDE6D O43924 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4686130 0.96 CCR5 (1.00) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544010 0.92 CCR5 (0.78) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL4682434 0.88 CCR5 (0.85) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL4740667 0.85 CCR5 (0.80) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544007 0.84 CCR5 (1.00) CCR5OPRM1OPRL1OPRD1OPRK1
SCHEMBL4682424 0.84 CCR5 (0.74) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL4683260 0.83 CCR5 (0.73) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL4683230 0.82 CCR5 (0.75) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544011 0.82 CCR5 (1.00) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL4680985 0.82 CCR5 (0.74) CCR5OPRM1OPRL1SLC6A9SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed