SCHEMBL13544010

SCHEMBL13544010

COc1cccc(N2CNC(=O)C23CCN(CCOC2(c4ccc(Cl)c(Cl)c4)CCN(C(=O)C4CCCC4)CC2)CC3)c1

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.78
OPRM1 P35372 5/20 0.46
OPRL1 P41146 5/20 0.46
SLC6A9 P48067 3/20 0.46
SLC6A5 Q9Y345 3/20 0.46
HTR1A P08908 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682434 0.96 CCR5 (0.85) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544006 0.92 CCR5 (0.92) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544013 0.90 CCR5 (0.66) CCR5OPRM1OPRL1
SCHEMBL4679294 0.87 CCR5 (0.68) CCR5OPRM1OPRL1
SCHEMBL4686130 0.87 CCR5 (1.00) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL14144448 0.86 CCR5 (0.64) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL13544009 0.85 CCR5 (0.85) CCR5OPRM1OPRL1HTR1AOPRD1
SCHEMBL4685629 0.84 CCR5 (0.64) CCR5OPRM1OPRL1
SCHEMBL14144443 0.84 CCR5 (0.62) CCR5OPRM1OPRL1SLC6A9SLC6A5
SCHEMBL6170250 0.83 CCR5 (0.63) CCR5OPRM1OPRL1HTR1AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed