SCHEMBL13544693

SCHEMBL13544693

CC(=O)c1c(F)ccc2[nH]c(N)nc12

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.44
HRH4 Q9H3N8 4/20 0.36
PNP P00491 2/20 0.36
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
KCNH2 Q12809 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PKM P14618 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
EGLN1 Q9GZT9 2/20 0.34
NUDT1 P36639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13544496 0.86 PARP1 (0.45) PARP1HRH4PNPCDK5CDK5R1
SCHEMBL13544691 0.83 PARP1 (0.45) PARP1HRH4PKMRXFP1EGLN1
SCHEMBL17276023 0.74 HRH4 (0.42) HRH4PNPCDK5CDK5R1EGLN1
SCHEMBL17276081 0.71 NUDT1 (0.49) PNPCDK5CDK5R1MAPTNPSR1
SCHEMBL13544692 0.71 PARP1 (0.41) PARP1PKMRXFP1EGLN1
SCHEMBL1193115 0.71 PARP1 (0.54) PARP1NUDT1
SCHEMBL13544493 0.70 PARP1 (0.45) PARP1HRH4EGLN1
SCHEMBL24112331 0.70 PKMYT1 (0.38) PARP1PNPCDK5CDK5R1
SCHEMBL1202101 0.70 CA12 (0.45) PARP1PNPCDK5CDK5R1PKM
SCHEMBL24112448 0.69 NUDT1 (0.40) PNPCDK5CDK5R1ALOX15KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed