SCHEMBL24112331

SCHEMBL24112331

CNC(=O)c1c(C)ccc2[nH]c(N)nc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKMYT1 Q99640 1/20 0.38
PIK3CA P42336 4/20 0.38
MTOR P42345 3/20 0.38
PNP P00491 2/20 0.38
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
FABP6 P51161 1/20 0.36
EGFR P00533 2/20 0.35
SRC P12931 1/20 0.35
KDM5A P29375 1/20 0.35
CYP1A2 P05177 1/20 0.34
MMP12 P39900 1/20 0.34
VCP P55072 1/20 0.34
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23835776 0.85 KDM4E (0.39) PIK3CAMTORPNPKDM5APARP1
SCHEMBL25808876 0.85 PKMYT1 (0.41) PKMYT1PIK3CAMTORPNPKDM5A
SCHEMBL24112448 0.84 NUDT1 (0.40) PNPCDK5CDK5R1PKN1PKN2
SCHEMBL24112332 0.75 PKN1 (0.61) PKN1PKN2PARP1
SCHEMBL2541920 0.72 CBFB (0.49) PNPCDK5CDK5R1FABP6MMP12
SCHEMBL6314907 0.71 PARP1 (0.36) PNPCDK5CDK5R1FABP6MMP12
SCHEMBL13544693 0.70 PARP1 (0.44) PNPCDK5CDK5R1PARP1
SCHEMBL1203243 0.70 ALDH1A1 (0.39) PNPPARP1
SCHEMBL24029084 0.70 PRKCZ (0.42) PKMYT1PNPKDM5AMMP12PARP1
SCHEMBL24450350 0.70 PRKCZ (0.42) PNPKDM5AMMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252644-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2021-12-16 WO disclosed