Nafamostat

Nafamostat

SCHEMBL135503

N=C(N)Nc1ccc(C(=O)Oc2ccc3cc(C(=N)N)ccc3c2)cc1

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 10/20 0.64
PLG P00747 9/20 0.64
F2 P00734 8/20 0.64
F12 P00748 6/20 0.64
KLK1 P06870 3/20 0.64
C1R P00736 2/20 0.64
F10 P00742 2/20 0.64
HGFAC Q04756 2/20 0.64
TMPRSS2 O15393 1/20 0.64
MLNR O43193 1/20 0.64
ALDH1A1 P00352 1/20 0.64
LMNA P02545 1/20 0.64
ITGB3 P05106 1/20 0.64
HPN P05981 1/20 0.64
CHRM2 P08172 1/20 0.64
ITGA2B P08514 1/20 0.64
C1S P09871 1/20 0.64
ADORA3 P0DMS8 1/20 0.64
MAPT P10636 1/20 0.64
CHRM1 P11229 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nafamostat SCHEMBL29429445 1.00 PRSS1 (0.64) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL29429443 1.00 PRSS1 (0.64) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL16069975 1.00 PRSS1 (0.64) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL3302794 0.99 PRSS1 (0.63) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL7345508 0.97 PRSS1 (0.62) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL874941 0.94 FTO (0.64) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL7051240 0.94 PLAU (0.58) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL1568755 0.94 FTO (0.70) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL564665 0.94 FTO (0.70) PRSS1PLGF2F12KLK1
Nafamostat SCHEMBL29832433 0.94 FTO (0.70) PRSS1PLGF2F12KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4150 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4228644-B1 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NANTCELL INC (US) 2026-05-27 EP claimed
US-12636253-B2 Modified release compositions of nafamostat and methods of using same Ensysce Biosciences Inc. (US) 2026-05-26 US claimed
US-20260139035-A1 HUMAN ANTIBODY AGAINST CORONAVIRUS VARIANTS OR ANTIGEN-BINDING FRAGMENT THEREOF NATIONAL UNIVERSITY CORPORATION KUMAMOTO UNIVERSITY (JP) 2026-05-21 US claimed
US-20260130921-A1 TREATMENT OF VIRAL INFECTIONS WITH COMBINATION OF PIKFYVE KINASE INHIBITORS AND TMPRSS-2 INHIBITORS AcuraStem Incorporated (US) 2026-05-14 US claimed
EP-4725496-A2 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NantCell, Inc. (US) 2026-04-15 EP claimed
US-12599578-B2 Compositions comprising enzyme-cleavable prodrugs and controlled release nafamostat and methods of use thereof Ensysce Biosciences Inc. (US) 2026-04-14 US claimed
US-12599644-B2 Treatment of coronavirus infection with Flt3 receptor interacting lectin (FRIL) ACADEMIA SINICA (TW) 2026-04-14 US claimed
US-20260007597-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRUS-INDUCED AIRWAY FIBROSIS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2026-01-08 US claimed
US-20250345458-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL INC (US) 2025-11-13 US claimed
US-20250332247-A1 IMPROVED CORONAVIRUS VACCINE ACADEMIA SINICA (TW) 2025-10-30 US claimed
EP-0647398-B1 ORGAN PRESERVING FLUID TORII PHARMACEUTICAL CO LTD (JP) 1997-09-17 EP claimed
US-5565317-A BIOLOGICAL ORGAN PRESERVATIVE; STORAGE STABILITY TORII PHARMACEUTICAL CO., LTD. (JP) 1996-10-15 US claimed
EP-0647398-A1 ORGAN PRESERVING FLUID TORII PHARMACEUTICAL CO., LTD (JP) 1995-04-12 EP claimed
EP-0287036-B1 NEW PHARMACEUTICAL COMPOSITIONS COMPRISING ESTERS OR AMIDES AS ACTIVE INGREDIENTS ONO PHARMACEUTICAL CO., LTD. (JP) 1991-04-10 EP claimed
US-4990537-A 6-amidinonaphth-2-yl or p-(n,n-dimethylcarbamoyl methoxy-carbonyl methyl) phenyl ester of p-guanidinobenzoic acid BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-02-05 US claimed
EP-0350840-A2 Antiviral agent BANYU PHARMACEUTICAL CO., LTD. (JP) 1990-01-17 EP claimed
EP-0287036-A2 New pharmaceutical compositions comprising esters or amides as active ingredients ONO PHARMACEUTICAL CO., LTD. (JP) 1988-10-19 EP claimed
EP-0048433-B1 NOVEL AMIDINE COMPOUNDS, PROCESS FOR PRODUCING SAME AND ANTI-COMPLEMENT AGENT COMPRISING THEM TORII & CO., LTD. (JP) 1986-05-28 EP claimed
US-4454338-A 6-AMIDINO-2-NATHTHYL-4-GUANIDINOBENZOATE TORII & CO., LTD. (JP) 1984-06-12 US claimed
EP-0048433-A2 Novel amidine compounds, process for producing same and anti-complement agent comprising them TORII & CO., LTD. (JP) 1982-03-31 EP claimed