Nafamostat

Nafamostat

SCHEMBL7051240

N=C(N)Nc1ccc(C(=O)Oc2ccc3cc(C(=N)N)ccc3c2)cc1.N=C(N)c1ccccc1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 8/20 0.58
PRSS1 P07477 9/20 0.58
F2 P00734 7/20 0.58
PLG P00747 7/20 0.58
F12 P00748 4/20 0.58
KLK1 P06870 3/20 0.58
MAPT P10636 2/20 0.58
C1R P00736 2/20 0.58
F10 P00742 2/20 0.58
TMPRSS2 O15393 1/20 0.58
MLNR O43193 1/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
ITGB3 P05106 1/20 0.58
HPN P05981 1/20 0.58
CHRM2 P08172 1/20 0.58
ITGA2B P08514 1/20 0.58
C1S P09871 1/20 0.58
ADORA3 P0DMS8 1/20 0.58
CHRM1 P11229 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nafamostat SCHEMBL7345508 0.94 PRSS1 (0.62) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL16069975 0.94 PRSS1 (0.64) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL135503 0.94 PRSS1 (0.64) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL29429443 0.94 PRSS1 (0.64) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL29429445 0.94 PRSS1 (0.64) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL3302794 0.93 PRSS1 (0.63) PLAUPRSS1F2PLGF12
SCHEMBL18720217 0.89 MAPT (0.61) PLAUPRSS1F2PLGF12
SCHEMBL7337750 0.89 F12 (0.71) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL1568755 0.88 FTO (0.70) PLAUPRSS1F2PLGF12
Nafamostat SCHEMBL874941 0.88 FTO (0.64) PLAUPRSS1F2PLGF12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003012450-A1 DIAGNOSTIC MARKERS OF LIVER DYSFUNCTION THE SCRIPPS RESEARCH INSTITUTE (US) 2003-02-13 WO disclosed