Rosoxacin

Rosoxacin

SCHEMBL135645

CCn1cc(C(=O)O)c(=O)c2ccc(-c3ccncc3)cc21

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.61
KDM4E B2RXH2 3/20 0.52
HPGD P15428 3/20 0.52
ALDH1A1 P00352 2/20 0.52
HSD17B10 Q99714 2/20 0.52
TSHR P16473 2/20 0.52
RAB9A P51151 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
APEX1 P27695 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
LMNA P02545 3/20 0.51
MEN1 O00255 1/20 0.51
ABCC4 O15439 1/20 0.51
PKM P14618 1/20 0.51
PTGS1 P23219 1/20 0.51
KMT2A Q03164 1/20 0.51
HTT P42858 1/20 0.51
ROCK2 O75116 4/20 0.49
CDK1 P06493 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rosoxacin SCHEMBL29361483 1.00 CAPN1 (0.61) CAPN1KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10475298 0.91 CAPN1 (0.59) CAPN1KDM4EHPGDALDH1A1HSD17B10
SCHEMBL11655148 0.90 CAPN1 (0.50) CAPN1KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10474600 0.89 CAPN1 (0.62) CAPN1ROCK2CDK1PRKACACDK2
SCHEMBL10475306 0.89 CAPN1 (0.57) CAPN1ROCK2CDK1PRKACACDK2
SCHEMBL10475297 0.88 CAPN1 (0.56) CAPN1
SCHEMBL11621910 0.87 LMNA (0.54) CAPN1KDM4EHPGDALDH1A1HSD17B10
SCHEMBL11620699 0.87 CAPN1 (0.58) CAPN1LMNAMEN1ABCC4PKM
SCHEMBL10475303 0.87 ROCK2 (0.63) CAPN1MEN1KMT2AROCK2CDK1
SCHEMBL10474604 0.87 ROCK2 (0.52) CAPN1KDM4EROCK2CDK1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4545 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4571306-A1 STABILIZING OXYGEN IN A COMPOSITION Instrumentation Laboratory Company (US) 2025-06-18 EP claimed
CN-120142412-A Stabilizing oxygen in a composition 仪器实验室公司 2025-06-13 CN claimed
US-20250189479-A1 STABILIZING OXYGEN IN A COMPOSITION INSTRUMENTATION LABORATORY COMPANY 2025-06-12 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4554939-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2025-05-21 EP claimed
EP-4554627-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-21 EP claimed
US-20250144088-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-08 US claimed
WO-2025080590-A1 CO-CRYSTALLIZATION OF ACTIVES WITH SACCHARIDE-BASED MOLECULAR FRAMEWORKS SCIENTIFIC HORIZONS CONSULTING LLC (US) 2025-04-17 WO claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-20250115942-A1 SCREENING METHOD FOR ANTI-PSEUDOMONAL AGENTS AND COMPOSITIONS AND METHODS FOR TREATING PSEUDOMONAS INFECTIONS BOARD OF REGENTS FOR THE OKLAHOMA AGRICULTURAL AND MECHANICAL COLLEGES 2025-04-10 US claimed
EP-0741570-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1996-11-13 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1995020387-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1995-08-03 WO claimed
WO-1991009616-A1 QUINOLONE ANTIBIOTICS ENCAPSULATED IN LIPID VESICLES YALE UNIVERSITY (US) 1991-07-11 WO claimed
US-4853225-A Process for implanting a medicament depot MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-08-01 US claimed
EP-0222814-A1 USE OF QUINOLONE DERIVATIVES FOR THE TREATMENT OF MYCOPLASMAL PNEUMONIA IN PIGS BEECHAM GROUP PLC (GB) 1987-05-27 EP claimed
WO-1986006630-A1 USE OF QUINOLONE DERIVATIVES FOR THE TREATMENT OF MYCOPLASMAL PNEUMONIA IN PIGS BEECHAM GROUP P.L.C. (GB) 1986-11-20 WO claimed
EP-0098577-A2 Drugs for treating diarrhea caused by infection HOECHST AKTIENGESELLSCHAFT (DE) 1984-01-18 EP claimed