SCHEMBL13565014

SCHEMBL13565014

CC(C)(C)S(=O)(=O)Nc1ccc(CNc2cccc3c2Cc2ccccc2-3)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36
PNMT P11086 1/20 0.34
AGTR2 P50052 1/20 0.34
METAP2 P50579 1/20 0.33
ITGA1 P56199 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
JAK2 O60674 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565712 0.84 NPC1 (0.43) NPC1RAB9ASMN1; SMN2HTTNPSR1
SCHEMBL11935308 0.83 HTT (0.56) SMN1; SMN2HTTNPSR1RXRARXRB
SCHEMBL10116309 0.79 NPC1 (0.54) NPC1RAB9AHTTNPSR1MAPT
SCHEMBL15671164 0.78 RAB9A (0.51) NPC1RAB9ASMN1; SMN2HTTNPSR1
SCHEMBL13565626 0.76 PSIP1 (0.44) HSD17B10HDAC6CA1CA2
SCHEMBL11935952 0.76 NPC1 (0.47) NPC1RAB9ASMN1; SMN2HTTNPSR1
SCHEMBL13564926 0.75 NPC1 (0.45) NPC1RAB9ASMN1; SMN2HTTNPSR1
SCHEMBL13565494 0.74 SCD (0.44)
SCHEMBL13564999 0.74 CA1 (0.50) HTTCA1CA2
SCHEMBL13565011 0.73 CA1 (0.53) SMN1; SMN2HTTMAPTHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed