SCHEMBL13565249

SCHEMBL13565249

CC1CCC(Oc2ccc(NCCCCCNS(=O)(=O)C(C)C)cc2)C1C

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 3/20 0.41
NPY5R Q15761 7/20 0.38
KDM1A O60341 1/20 0.33
HTR1A P08908 1/20 0.33
KCNH2 Q12809 3/20 0.32
HRH1 P35367 2/20 0.32
CNR2 P34972 1/20 0.31
GRIA4 P48058 1/20 0.30
ALDH1A1 P00352 2/20 0.30
PKM P14618 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565287 0.85 CNR2 (0.35) CNR2ALDH1A1PKMUSP2
SCHEMBL10115508 0.85 ALDH1A1 (0.42) HTR1AALDH1A1PKMUSP2
SCHEMBL11935821 0.82 GRIA1 (0.45) GRIA1NPY5RKCNH2HRH1ALDH1A1
SCHEMBL13565799 0.81 GRIA1 (0.44) GRIA1NPY5RKCNH2HRH1ALDH1A1
SCHEMBL11935717 0.80 GAA (0.37)
SCHEMBL13565895 0.80 GRIA1 (0.45) GRIA1NPY5RKCNH2CNR2
SCHEMBL13565487 0.79 GRIA1 (0.42) GRIA1NPY5RKDM1AGRIA4
SCHEMBL13565144 0.79 CTSL (0.44) GRIA1NPY5RKCNH2HRH1
SCHEMBL11936141 0.78 HRH3 (0.41) ALDH1A1
SCHEMBL11935850 0.78 GRIA1 (0.41) GRIA1NPY5RKDM1AHTR1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed