SCHEMBL13565320

SCHEMBL13565320

CCCN1C(=O)c2ccc(NCCCCCNS(=O)(=O)C(C)(C)C)cc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
HPGD P15428 4/20 0.40
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 2/20 0.40
BRD4 O60885 1/20 0.39
MAPK1 P28482 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
DNMT1 P26358 1/20 0.38
DNMT3L Q9UJW3 1/20 0.38
DNMT3A Q9Y6K1 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 3/20 0.38
CNR2 P34972 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RGS12 O14924 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565336 0.91 POLB (0.39) ALDH1A1HPGDKDM4EHSD17B10BRD4
SCHEMBL13564882 0.89 CNR2 (0.44) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL13439076 0.86 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL10115058 0.84 ALDH1A1 (0.56) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL13565192 0.83 CNR2 (0.34) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL17090230 0.82 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL13565702 0.81 ESR1 (0.40) ALDH1A1HPGDKDM4EMAPK1MEN1
SCHEMBL11935601 0.81 ALDH1A1 (0.48) ALDH1A1HPGDHSD17B10MAPK1MEN1
SCHEMBL11935610 0.81 ALDH1A1 (0.44) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL11935602 0.81 ALDH1A1 (0.39) ALDH1A1HPGDKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed