SCHEMBL13565448

SCHEMBL13565448

CCc1cccc(CCCNCC2CCC(NS(=O)(=O)C(C)(C)C)CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.38
CXCR4 P61073 2/20 0.36
TP53 P04637 2/20 0.36
LMNA P02545 2/20 0.36
POLB P06746 2/20 0.36
MAPT P10636 1/20 0.35
FKBP1A P62942 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565454 0.88 LMNA (0.38) TP53LMNAPOLBMAPTALDH1A1
SCHEMBL17090086 0.84 POLB (0.44) POLBMAPTALDH1A1
SCHEMBL13564861 0.84 POLB (0.44) POLBMAPTALDH1A1
SCHEMBL10114161 0.84 NPY5R (0.43) TP53LMNAPOLBFKBP1AALDH1A1
SCHEMBL13565579 0.83 SCN8A (0.38)
SCHEMBL13565419 0.81 MEN1 (0.46) TP53LMNAPOLBMAPTALDH1A1
SCHEMBL13565543 0.81 KMT2A (0.46) POLBALDH1A1
SCHEMBL11935165 0.78 SMYD3 (0.50) SMYD3CXCR4
SCHEMBL13564840 0.77 CNR1 (0.38) MAPT
SCHEMBL13565548 0.77 CNR2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed