SCHEMBL13565660

SCHEMBL13565660

CC(C)S(=O)(=O)NCCCCCNc1ccc2c(c1)C(=O)N(c1ccc(C(F)(F)F)cc1)C2=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 5/20 0.39
CA1 P00915 4/20 0.39
CA12 O43570 3/20 0.39
CA2 P00918 3/20 0.39
GRIA1 P42261 3/20 0.38
POLB P06746 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.35
GRIA4 P48058 1/20 0.35
NPY5R Q15761 1/20 0.35
CA4 P22748 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HPSE Q9Y251 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13566071 0.90 ALDH1A1 (0.48) CA9CA1CA12CA2GRIA1
SCHEMBL13566016 0.88 GRIA1 (0.40) CA9CA1CA12CA2GRIA1
SCHEMBL11935357 0.88 GRIA1 (0.41) GRIA1POLBALDH1A1HPGDMAPT
SCHEMBL10115535 0.87 ALDH1A1 (0.43) POLBALDH1A1HPGDMEN1KMT2A
SCHEMBL13565962 0.87 CA9 (0.42) CA9CA1CA12CA2POLB
SCHEMBL13566094 0.85 GRIA1 (0.37) CA9CA1CA12CA2GRIA1
SCHEMBL13565723 0.85 GRIA1 (0.40) CA9CA1CA12CA2GRIA1
SCHEMBL11935719 0.82 ALDH1A1 (0.40) CA9CA1CA12CA2POLB
SCHEMBL17090278 0.82 GRIA1 (0.46) GRIA1POLBALDH1A1HPGDNPY5R
SCHEMBL13565051 0.81 GRIA1 (0.54) CA1CA2GRIA1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed