SCHEMBL13565962

SCHEMBL13565962

CC(C)(C)S(=O)(=O)NCCCCCNc1ccc2c(c1)C(=O)N(c1ccc(C(F)(F)F)cc1)C2=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 5/20 0.42
CA12 O43570 3/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
POLB P06746 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.36
CNR2 P34972 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HPSE Q9Y251 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11935601 0.91 ALDH1A1 (0.48) CA9CA12CA1CA2POLB
SCHEMBL13565702 0.89 ESR1 (0.40) CA9CA12CA1CA2POLB
SCHEMBL11935602 0.88 ALDH1A1 (0.39) CA9CA12CA1CA2POLB
SCHEMBL13565967 0.87 ALDH1A1 (0.38) CA9CA12CA1CA2POLB
SCHEMBL13565660 0.87 CA9 (0.39) CA9CA12CA1CA2POLB
SCHEMBL10115349 0.87 ALDH1A1 (0.43) CA9CA12CA1CA2POLB
SCHEMBL11935719 0.83 ALDH1A1 (0.40) CA9CA12CA1CA2POLB
SCHEMBL13564882 0.82 CNR2 (0.44) POLBALDH1A1HPGDMAPTCNR2
SCHEMBL11935312 0.81 MAPT (0.43) CA1CA2POLBMAPTCNR2
SCHEMBL17090252 0.81 CA1 (0.41) CA9CA12CA1CA2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed