SCHEMBL13565993

SCHEMBL13565993

CC(C)S(=O)(=O)Nc1ccc(CNc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.55
FFAR1 O14842 1/20 0.52
KIF11 P52732 4/20 0.48
ADRA2A P08913 1/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA12 O43570 1/20 0.45
CA7 P43166 1/20 0.45
CACNA1B Q00975 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.42
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11936113 0.90 PPARA (0.56) PPARAFFAR1KIF11CA1CA2
SCHEMBL13565306 0.87 CA1 (0.62) CA1CA2
SCHEMBL13565690 0.86 PPARA (0.46) PPARAFFAR1ALDH1A1
SCHEMBL13565986 0.85 CA1 (0.49) PPARACA1CA2
SCHEMBL13565070 0.85 PPARA (0.50) PPARAFFAR1KIF11ADRA2ACA1
SCHEMBL13565065 0.84 KDM4E (0.44) FFAR1CA1CA2CA12CA7
SCHEMBL13565366 0.84 PPARA (0.49) PPARAKIF11ALDH1A1
SCHEMBL10116639 0.83 PPARA (0.67) PPARA
SCHEMBL13565877 0.83 HDAC1 (0.55) PPARAKIF11CA1CA2CA12
SCHEMBL13566019 0.82 CA1 (0.50) FFAR1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed