SCHEMBL13565877

SCHEMBL13565877

CC(C)S(=O)(=O)Nc1ccc(CNc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.55
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC7 Q8WUI4 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC9 Q9UKV0 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
KIF11 P52732 1/20 0.50
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA7 P43166 1/20 0.48
HTT P42858 2/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11936062 0.84 CA1 (0.62) CA12CA1CA2CA7HTT
SCHEMBL13565924 0.83 HDAC1 (0.56) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL13565993 0.83 PPARA (0.55) KIF11CA12CA1CA2CA7
SCHEMBL13565235 0.82 HPGD (0.54) CA12CA1CA2CA7HTT
SCHEMBL13565270 0.82 HDAC3 (0.38) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL13565065 0.81 KDM4E (0.44) CA12CA1CA2CA7MAPT
SCHEMBL4182657 0.80 ALDH1A1 (0.59) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL17090488 0.79 LMNA (0.54) CA12CA1CA2HTTMEN1
SCHEMBL13566019 0.79 CA1 (0.50) CA12CA1CA2HTTMEN1
SCHEMBL13565984 0.79 CA1 (0.59) CA12CA1CA2CA7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed