SCHEMBL13575481

SCHEMBL13575481

COc1cc(C(=O)NC2CCN(C3CC3)CC2)ccc1N

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.52
KMT2A Q03164 1/20 0.49
HTR4 Q13639 1/20 0.49
MCHR1 Q99705 2/20 0.48
ACHE P22303 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
IGF1R P08069 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12389339 0.95 F10 (0.58) F10KMT2AHTR4CYP2D6CYP2C9
SCHEMBL13461288 0.93 SLC6A5 (0.51) F10KMT2AHTR4
SCHEMBL13881274 0.92 F10 (0.60) F10KMT2AHTR4MCHR1IGF1R
SCHEMBL12893788 0.91 HTR4 (0.48) F10KMT2AHTR4MCHR1CYP2D6
SCHEMBL12894062 0.91 HTR4 (0.48) F10KMT2AHTR4MCHR1CYP2D6
SCHEMBL13881189 0.90 KMT2A (0.57) F10KMT2AHTR4CYP2D6CYP2C9
SCHEMBL736450 0.90 KMT2A (0.57) F10KMT2AHTR4CYP2D6CYP2C9
SCHEMBL13181455 0.90 KMT2A (0.57) F10KMT2AHTR4CYP2D6CYP2C9
SCHEMBL13457659 0.89 HTR4 (0.52) F10HTR4MCHR1ACHE
SCHEMBL12893438 0.88 HTR4 (0.52) F10KMT2AHTR4MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009153197-A1 HALO-SUBSTITUTED PYRIMIDODIAZEPINES AS PLKL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-12-23 WO disclosed