SCHEMBL13575643

SCHEMBL13575643

Bc1cnc2n1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.47
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
ESR2 Q92731 1/20 0.40
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
PDK2 Q15119 1/20 0.40
GPR119 Q8TDV5 4/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.38
ATM Q13315 1/20 0.38
USP2 O75604 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17790245 0.85 P2RX7 (0.48) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL17788667 0.84 NR1H2 (0.45) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL10007648 0.84 P2RX7 (0.51) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL31568967 0.84 P2RX7 (0.47) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL10183072 0.84 NR1H2 (0.47) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL601417 0.84 P2RX7 (0.47) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL19005602 0.83 NR1H2 (0.46) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL31569288 0.83 NR1H2 (0.46) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL28887447 0.83 NR1H2 (0.49) NR1H2MAPTPOLBESR2CKS1B
SCHEMBL10235383 0.82 NR1H2 (0.45) NR1H2MAPTPOLBESR2CKS1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158394-A1 DIKETO AZOLOPIPERIDINES AND AZOLOPIPERAZINES AS ANTI-HIV AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-12-30 WO disclosed