SCHEMBL13605156

SCHEMBL13605156

COc1cc2nccc(Oc3ccc(C)nc3C(=O)c3ccccc3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SRC P12931 5/20 0.69
TGFBR1 P36897 5/20 0.69
PDGFRA P16234 4/20 0.52
FGFR2 P21802 2/20 0.52
KDR P35968 1/20 0.52
MET P08581 4/20 0.50
KIT P10721 2/20 0.50
PDGFRB P09619 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3892904 0.90 SRC (0.58) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL13605158 0.86 SRC (0.54) SRCTGFBR1PDGFRAKDRMET
SCHEMBL3896433 0.85 SRC (0.66) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL3907600 0.85 SRC (0.68) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL3903245 0.82 SRC (1.00) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL3894063 0.81 SRC (1.00) SRCTGFBR1PDGFRAFGFR2KDR
Hydrochloric Acid SCHEMBL3896851 0.81 SRC (1.00) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL13605034 0.81 SRC (0.78) SRCTGFBR1PDGFRAFGFR2KDR
Hydrochloric Acid SCHEMBL3908414 0.80 SRC (0.98) SRCTGFBR1PDGFRAFGFR2KDR
SCHEMBL7487378 0.80 FGFR2 (0.77) SRCTGFBR1PDGFRAFGFR2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090312313-A1 COMPOUND HAVING TGFBETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2009-12-17 US disclosed
US-20090312313-A1 COMPOUND HAVING TGFBETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2009-12-17 US disclosed
US-7560558-B2 Compound having TGFβ inhibitory activity and medicinal composition containing the same KIRIN BEER KABUSHIKI KAISHA (JP) 2009-07-14 US disclosed
US-7560558-B2 Compound having TGFβ inhibitory activity and medicinal composition containing the same KIRIN BEER KABUSHIKI KAISHA (JP) 2009-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312313-A1 COMPOUND HAVING TGFBETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME TGFB1, TGFBR1, TGFBR2 SRC 496/4885TGFBR1 2/4885PDGFRA 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.