SCHEMBL13610427

SCHEMBL13610427

O=CN1CCC2(CC1)OC(=O)c1cc(F)ccc12

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 8/20 0.57
NPY5R Q15761 9/20 0.49
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14349499 0.83 AVPR1A (0.60) AVPR1ANPY5RSIGMAR1
SCHEMBL2359969 0.80 SIGMAR1 (0.73) AVPR1ASIGMAR1
SCHEMBL738397 0.77 AVPR1A (0.50) AVPR1ANPY5RSIGMAR1
Hydrochloric Acid SCHEMBL6820620 0.76 AVPR1A (0.49) AVPR1ANPY5RSIGMAR1
SCHEMBL4577444 0.76 AVPR1A (0.58) AVPR1ANPY5R
SCHEMBL30136877 0.74 AVPR1A (1.00) AVPR1A
SCHEMBL16836272 0.74 AVPR1A (1.00) AVPR1A
SCHEMBL6054773 0.73 AVPR1A (0.54) AVPR1ANPY5R
SCHEMBL4367569 0.72 AVPR1A (0.48) AVPR1ANPY5RSIGMAR1
SCHEMBL1998588 0.72 NPY5R (0.48) AVPR1ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629353-B2 Indol-3-yl-carbonyl-spiro-piperidine derivatives as V1a receptor antagonists HOFFMAN-LA ROCHE INC. (US) 2009-12-08 US disclosed