SCHEMBL13613342

SCHEMBL13613342

NC(=O)C(N)c1ccc(F)cc1[N+](=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.34
CES1 P23141 4/20 0.34
TDP1 Q9NUW8 2/20 0.33
ATM Q13315 1/20 0.33
PARP1 P09874 1/20 0.33
DPP9 Q86TI2 1/20 0.32
KEAP1 Q14145 1/20 0.32
GRM1 Q13255 2/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
KMT2A Q03164 1/20 0.31
PDE7A Q13946 1/20 0.31
EPHX1 P07099 1/20 0.31
KCNN4 O15554 4/20 0.30
KCNMA1 Q12791 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1115202 0.78 CES2 (0.50) CES2CES1PARP1DPP9KEAP1
Hydrochloric Acid SCHEMBL3620524 0.72 DPP4 (0.43) CES2CES1ATMPARP1KMT2A
Hydrochloric Acid SCHEMBL3620520 0.72 DPP4 (0.43) CES2CES1ATMPARP1KMT2A
SCHEMBL13613341 0.71 TSHR (0.37) TDP1PARP1GRM1MEN1CYP1A2
Hydrochloric Acid SCHEMBL4563584 0.68 DPP4 (0.45) TDP1GRM1MEN1CYP1A2KMT2A
SCHEMBL17347338 0.67 ATM (0.65) CES2CES1TDP1ATMALDH1A1
SCHEMBL3831033 0.66 TDP1 (0.41) TDP1ATMPARP1PDE7AKCNMA1
SCHEMBL5114349 0.65 HDAC3 (0.45) CES2CES1EPHX1KCNN4ALDH1A1
SCHEMBL5114354 0.65 HDAC3 (0.45) CES2CES1EPHX1KCNN4ALDH1A1
SCHEMBL6321555 0.65 HDAC3 (0.45) CES2CES1EPHX1KCNN4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119703-A1 NOVEL INDOLE DERIVATIVE HAVING INHIBITORY ACTIVITY ON I B KINASE Santen Pharmaceutical Co., Ltd (JP) 2009-11-18 EP disclosed