SCHEMBL13615436

SCHEMBL13615436

CCC(=O)c1cccc(-c2ccc3nc(NC(C)=O)sc3c2)c1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 8/20 0.70
PIK3CA P42336 5/20 0.64
RAB9A P51151 2/20 0.58
ABL1 P00519 1/20 0.57
CYP3A4 P08684 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.56
NPC1 O15118 1/20 0.56
STAT1 P42224 1/20 0.56
DYRK1A Q13627 3/20 0.55
SMO Q99835 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798579 0.88 PIK3CG (0.77) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2
SCHEMBL3711448 0.86 DYRK1A (0.75) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2
SCHEMBL1651716 0.86 SMN1; SMN2 (0.75) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2
SCHEMBL3709415 0.85 PIK3CG (0.76) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2
SCHEMBL1651874 0.83 PIK3CG (1.00) PIK3CGPIK3CARAB9AABL1CYP3A4
SCHEMBL3714360 0.83 PIK3CG (0.65) PIK3CGPIK3CAABL1CYP3A4SMN1; SMN2
SCHEMBL3716998 0.82 PIK3CG (0.79) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2
SCHEMBL1651394 0.82 PIK3CG (0.79) PIK3CGPIK3CARAB9AABL1CYP3A4
SCHEMBL3870265 0.82 PIK3CG (0.79) PIK3CGPIK3CARAB9AABL1CYP3A4
SCHEMBL1622337 0.81 PIK3CG (0.77) PIK3CGPIK3CARAB9ACYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133127-A1 FUSED BICYCLIC COMPOUNDS AND USE THEREOF AS PI3K INHIBITORS MERCK SERONO S.A. (CH) 2009-11-05 WO disclosed