SCHEMBL3714360

SCHEMBL3714360

CC(=O)Nc1nc2ccc(-c3cccc(C(=O)NCCO)c3)cc2s1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 5/20 0.65
PIK3CA P42336 5/20 0.59
SMN1; SMN2 Q16637 1/20 0.57
SMO Q99835 2/20 0.56
ABL1 P00519 3/20 0.53
CYP3A4 P08684 1/20 0.53
PKM P14618 1/20 0.52
PTGES O14684 1/20 0.52
DYRK1A Q13627 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1651716 0.87 SMN1; SMN2 (0.75) PIK3CGPIK3CASMN1; SMN2SMOCYP3A4
SCHEMBL798579 0.84 PIK3CG (0.77) PIK3CGPIK3CASMN1; SMN2SMOCYP3A4
SCHEMBL13615436 0.83 PIK3CG (0.70) PIK3CGPIK3CASMN1; SMN2SMOABL1
SCHEMBL3711448 0.82 DYRK1A (0.75) PIK3CGPIK3CASMN1; SMN2SMOCYP3A4
SCHEMBL3709415 0.81 PIK3CG (0.76) PIK3CGPIK3CASMN1; SMN2CYP3A4DYRK1A
SCHEMBL13188175 0.80 PIK3CG (0.64) PIK3CGPIK3CACYP3A4
SCHEMBL1651874 0.79 PIK3CG (1.00) PIK3CGPIK3CASMN1; SMN2ABL1CYP3A4
SCHEMBL3716998 0.79 PIK3CG (0.79) PIK3CGPIK3CASMN1; SMN2CYP3A4DYRK1A
SCHEMBL1651394 0.79 PIK3CG (0.79) PIK3CGPIK3CASMN1; SMN2ABL1CYP3A4
SCHEMBL3870265 0.79 PIK3CG (0.79) PIK3CGPIK3CASMN1; SMN2ABL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed