SCHEMBL13616448

SCHEMBL13616448

CCCc1cc(Br)cc(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.47
CYP19A1 P11511 1/20 0.43
CALM1 P0DP23 5/20 0.41
AKR1B1 P15121 1/20 0.41
ALDH1A1 P00352 2/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
MAOB P27338 2/20 0.38
CYP3A4 P08684 1/20 0.37
DAO P14920 1/20 0.37
PTPN1 P18031 1/20 0.36
NOS2 P35228 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10473733 0.85 PTGS2 (0.63) PTGS2CYP3A4
SCHEMBL10472797 0.85 PTGS2 (0.63) PTGS2CYP3A4
SCHEMBL427550 0.85 CYP19A1 (0.55) PTGS2CYP19A1CALM1AKR1B1ALDH1A1
SCHEMBL12044476 0.83 PTGS2 (0.43) PTGS2CYP19A1CALM1AKR1B1ALDH1A1
SCHEMBL2424239 0.82 TAAR1 (0.55) CYP19A1MAOBTAAR1
SCHEMBL10472749 0.82 PTGS2 (0.39) PTGS2CYP19A1CALM1AKR1B1ALDH1A1
SCHEMBL18854254 0.80 POLB (0.38) PTGS2ALDH1A1CYP3A4TAAR1
SCHEMBL11819334 0.80 IDO1 (0.41) PTGS2ALDH1A1CYP3A4TAAR1
SCHEMBL13980912 0.79 PTGS2 (0.50) PTGS2CYP19A1CALM1AKR1B1ALDH1A1
SCHEMBL29774677 0.79 ALDH1A1 (0.42) CYP19A1CALM1AKR1B1ALDH1A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015196335-A1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF TOCOPHERX, INC. (US) 2015-12-30 WO disclosed
WO-2014058747-A1 5-PHENOXY-3H-PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS HIV REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-04-17 WO disclosed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed