SCHEMBL13617452

SCHEMBL13617452

CSC(=O)C1=C(c2cccc(O)c2)CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.51
NR1H2 P55055 1/20 0.42
ABL1 P00519 1/20 0.41
EGFR P00533 1/20 0.41
SRC P12931 1/20 0.41
ABL2 P42684 1/20 0.41
MAPK1 P28482 1/20 0.38
NAMPT P43490 1/20 0.38
UCHL1 P09936 1/20 0.37
GRM5 P41594 2/20 0.37
KDM1A O60341 1/20 0.37
C5AR1 P21730 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
F12 P00748 1/20 0.36
PDK4 Q16654 1/20 0.36
USP30 Q70CQ3 2/20 0.36
PARP1 P09874 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8264285 0.88 ESR2 (0.54) ESR2NR1H2ABL1EGFRSRC
SCHEMBL8253723 0.86 ESR2 (0.52) ESR2NR1H2ABL1EGFRSRC
SCHEMBL8264299 0.82 ESR2 (0.47) ESR2NR1H2ABL1EGFRSRC
SCHEMBL8264160 0.78 USP30 (0.47) ESR2NR1H2MAPK1UCHL1PDK4
SCHEMBL8264380 0.77 ESR2 (0.49) ESR2NR1H2NAMPTUSP30PTPN2
SCHEMBL8265146 0.76 ESR2 (0.45) ESR2NR1H2MAPK1NAMPTUCHL1
SCHEMBL13490542 0.76 ESR2 (0.45) ESR2NR1H2MAPK1UCHL1HDAC1
SCHEMBL7047941 0.76 SLC6A3 (0.47) ESR2NR1H2MAPK1UCHL1USP30
SCHEMBL951850 0.76 ESR2 (0.48) ESR2NR1H2MAPK1NAMPTUCHL1
SCHEMBL8261717 0.75 CHRM2 (0.51) ESR2NR1H2MAPK1NAMPTUCHL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed