SCHEMBL13618728

SCHEMBL13618728

Cn1nc(C(C)(C)C)cc1-c1nnc(C(C)(C)[SH](C)(=O)Cc2ccc(F)cc2)[nH]1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPK14 Q16539 7/20 0.32
KDM4E B2RXH2 1/20 0.32
GRN P28799 1/20 0.32
SORT1 Q99523 1/20 0.32
GAA P10253 1/20 0.32
ERBB2 P04626 1/20 0.31
MAPK11 Q15759 1/20 0.31
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL350932 0.80 ALDH1A1 (0.35) ALDH1A1MAPTMAPK1NPSR1MAPK14
SCHEMBL10147492 0.79 ALDH1A1 (0.34) ALDH1A1MAPTMAPK1NPSR1MAPK14
SCHEMBL13618729 0.78
SCHEMBL351873 0.77 CNR2 (0.39) ALDH1A1MAPTMAPK14KDM4EGRN
SCHEMBL10146074 0.74 KDM4E (0.42) MAPTMAPK14KDM4EGRNSORT1
SCHEMBL13618716 0.71 KDM4E (0.40) MAPTMAPK14KDM4EGRNSORT1
SCHEMBL10147819 0.67 KDM4E (0.42) MAPTMAPK14KDM4EGRNSORT1
SCHEMBL351120 0.66 CNR2 (0.51) MAPTMAPK14KDM4EGRNSORT1
SCHEMBL12747060 0.66 KDM4E (0.41) MAPTMAPK14KDM4EGRNSORT1
SCHEMBL352612 0.65 KDM4E (0.33) KDM4EGRNSORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140089-A2 SULFONE COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-11-19 WO disclosed