SCHEMBL13620099

SCHEMBL13620099

O=Nc1cccc(C(=O)c2cc(F)ccc2F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.47
CES1 P23141 4/20 0.47
MDM2 Q00987 3/20 0.39
PARP1 P09874 1/20 0.38
MAPK14 Q16539 2/20 0.37
CTSL P07711 2/20 0.36
CTSK P43235 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL333382 0.79 CES2 (0.59) CES2CES1MAPK14HDAC1MEN1
SCHEMBL29367263 0.79 CES2 (0.59) CES2CES1MAPK14HDAC1MEN1
SCHEMBL4537134 0.75 CES2 (0.63) CES2CES1MDM2HDAC1MEN1
SCHEMBL27673772 0.74 CES2 (0.74) CES2CES1MDM2MEN1KMT2A
SCHEMBL12196344 0.74 CES2 (0.55) CES2CES1MEN1KMT2ANPC1
SCHEMBL9037143 0.72 LTA4H (0.61) CES2CES1MAPK14MEN1KMT2A
SCHEMBL2860775 0.72 KDM4E (0.51) CES2CES1PARP1HDAC1HDAC6
SCHEMBL8606277 0.71 ATM (0.52) MAPK14CTSLCTSKMEN1KMT2A
SCHEMBL9766594 0.71 ATM (0.52) MAPK14CTSLCTSKMEN1KMT2A
SCHEMBL20158111 0.70 CES2 (0.57) CES2CES1MDM2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009132832-A2 METHOD FOR THE PRODUCTION OF 1,4-BENZOTHIEPIN-1,1-DIOXIDE DERIVATIVES SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2009-11-05 WO disclosed