SCHEMBL13620294

SCHEMBL13620294

C=C(N1CCN(c2ccc(C(F)(F)F)cc2)CC1)C1(NC(=O)CC(c2ccccc2)c2ccccc2)CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 3/20 0.45
CACNB1 Q02641 3/20 0.45
CACNA1A O00555 2/20 0.45
CACNA1B Q00975 2/20 0.45
CACNA1C Q13936 2/20 0.45
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
CA12 O43570 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
AKR1C3 P42330 1/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 3/20 0.40
TACR1 P25103 2/20 0.40
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
MAPK1 P28482 1/20 0.39
SLC6A9 P48067 1/20 0.39
LDHA P00338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4456715 0.91 LMNA (0.53) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL13620516 0.88 LMNA (0.45) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL4248134 0.80 LMNA (0.64) LMNATSHR
SCHEMBL4453428 0.80 TSHR (0.56) CACNA2D1CACNB1CACNA1BCACNA1CLMNA
SCHEMBL13620078 0.78 LMNA (0.57) LMNATSHR
SCHEMBL13671111 0.78 LMNA (0.54) LMNATSHR
SCHEMBL13671109 0.78 LMNA (0.56) CACNA2D1CACNB1CACNA1BCACNA1CLMNA
SCHEMBL4450270 0.78 LMNA (0.56) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL4456969 0.74 TSHR (0.51) LMNATSHR
SCHEMBL4453699 0.74 LMNA (0.53) LMNATSHRCYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009132452-A1 DIARYL-CYCLYLALKYL DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2009-11-05 WO disclosed