SCHEMBL13620467

SCHEMBL13620467

Fc1ccc(/C=C/c2nc3ccc(C4=CCCO4)cc3o2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 5/20 0.39
METAP2 P50579 2/20 0.34
NR3C2 P08235 2/20 0.32
ROCK2 O75116 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
KCNH2 Q12809 1/20 0.31
SNCA P37840 1/20 0.31
GPR119 Q8TDV5 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP2D6 P10635 1/20 0.30
HPGD P15428 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13620319 0.90 METAP2 (0.44) NFE2L2METAP2HDAC6SNCAGPR119
SCHEMBL4062300 0.79 NFE2L2 (0.48) NFE2L2HTR2AHTR2CKCNH2KDM4E
SCHEMBL4062306 0.79 NFE2L2 (0.48) NFE2L2HTR2AHTR2CKCNH2KDM4E
SCHEMBL4051608 0.75 NFE2L2 (0.40) NFE2L2GPR119
SCHEMBL4051602 0.75 NFE2L2 (0.40) NFE2L2GPR119
SCHEMBL4057657 0.74 NFE2L2 (0.44) NFE2L2NR3C2HDAC6PTGS1PTGS2
SCHEMBL4057664 0.74 NFE2L2 (0.44) NFE2L2NR3C2HDAC6PTGS1PTGS2
SCHEMBL23064075 0.74 NFE2L2 (0.54) NFE2L2HDAC6PTGS1PTGS2HTR2A
SCHEMBL26327019 0.74 NFE2L2 (0.54) NFE2L2HDAC6PTGS1PTGS2HTR2A
SCHEMBL4054688 0.71 METAP2 (0.44) NFE2L2METAP2GPR119KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed