SCHEMBL13620559

SCHEMBL13620559

FC(F)(F)c1cc(-c2nc3ccc(C4=CCCO4)cc3o2)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.40
S1PR1 P21453 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13620439 0.93 TLR9 (0.40) TLR9S1PR1HDAC6HDAC3HDAC1
SCHEMBL4057433 0.74 S1PR1 (0.43) TLR9S1PR1HDAC6HDAC3HDAC1
SCHEMBL4054203 0.73 GPR119 (0.49) TLR9NPC1RAB9AESR1ESR2
SCHEMBL4050496 0.73 VSIR (0.53) TLR9HDAC6HDAC3HDAC1HDAC8
SCHEMBL18935939 0.70 TLR9 (0.55) TLR9HDAC6HDAC3HDAC1HDAC2
SCHEMBL24038196 0.68 ESR1 (0.46) TLR9HDAC6HDAC3HDAC1HDAC2
SCHEMBL4051906 0.68 VSIR (0.50) TLR9HDAC6HDAC3HDAC1HDAC8
SCHEMBL4057037 0.68 HDAC6 (0.41) TLR9S1PR1HDAC6HDAC3HDAC1
SCHEMBL24038396 0.68 NPC1 (0.56) TLR9NPC1RAB9AESR1ESR2
SCHEMBL4059341 0.68 GPR119 (0.43) TLR9NPC1RAB9AESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed