SCHEMBL13622956

SCHEMBL13622956

CCCc1ccc(-c2nc(N)ns2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA2B P29275 2/20 0.47
ADORA1 P30542 2/20 0.47
SREBF2 Q12772 4/20 0.38
PIK3CA P42336 6/20 0.35
PI4KA P42356 5/20 0.35
PI4KB Q9UBF8 5/20 0.35
PIK3CD O00329 4/20 0.35
PIK3CB P42338 4/20 0.35
PIK3CG P48736 3/20 0.35
CYP19A1 P11511 1/20 0.35
HEXA P06865 1/20 0.35
HEXB P07686 1/20 0.35
PIK3C3 Q8NEB9 1/20 0.34
PIM1 P11309 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13629967 0.88 ADORA3 (0.50) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL13615797 0.81 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL20390358 0.80 ADORA3 (0.59) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL3657653 0.79 ADORA3 (0.47) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL12681394 0.76 ADORA3 (0.54) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL12680080 0.74 ADORA3 (0.51) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL15071926 0.73 ADORA3 (0.50) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL20391019 0.73 ADORA3 (0.62) ADORA3ADORA2AADORA2BADORA1PIK3CA
SCHEMBL20390356 0.72 SREBF2 (0.50) SREBF2ALDH1A1MAPTATML3MBTL1
SCHEMBL18822208 0.70 PRMT5 (0.41) PIK3CAPI4KAPI4KBPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137737-A2 ANTI-BACTERIAL ACTIVITY OF 9-HYDROXY DERIVATIVES OF 6, 11-BICYCLOLIDES ENANTA PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed