SCHEMBL13623787

SCHEMBL13623787

COc1ccc(N)cc1C(=O)c1ncc(Cl)cc1NS(=O)(=O)c1ccc(C)c(CF)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.41
ALDH1A1 P00352 4/20 0.40
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CCR2 P41597 5/20 0.40
CYP3A4 P08684 5/20 0.40
CYP2C19 P33261 3/20 0.40
CCR4 P51679 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CCR5 P51681 1/20 0.40
HTT P42858 2/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306059 0.87 CYP2C9 (0.51) CYP2C9ALDH1A1TP53SMN1; SMN2CCR2
SCHEMBL306862 0.82 CYP2C9 (0.60) CYP2C9CCR2CYP3A4
SCHEMBL12594683 0.79 CCR2 (0.49) CYP2C9ALDH1A1TP53CCR2CYP3A4
SCHEMBL13623790 0.79 CCR2 (0.39) CYP2C9ALDH1A1TP53CCR2CYP3A4
SCHEMBL10272350 0.78 CYP2C9 (0.53) CYP2C9CCR2CYP3A4CYP2C19CCR4
SCHEMBL10272290 0.78 CYP3A4 (0.63) CYP2C9CCR2CYP3A4CYP2C19CCR4
SCHEMBL12594353 0.78 MEN1 (0.50) CYP2C9CCR2CYP3A4CYP2C19CCR4
SCHEMBL12593734 0.77 CYP2C9 (0.56) CYP2C9CCR2CYP3A4
SCHEMBL307207 0.76 CYP2C9 (0.48) CYP2C9ALDH1A1TP53CCR2CYP3A4
SCHEMBL10223328 0.76 CCR2 (0.57) CYP2C9ALDH1A1SMN1; SMN2CCR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622583-B2 Heteroaryl sulfonamides and CCR2 CHEMOCENTRYX, INC. (US) 2009-11-24 US disclosed