SCHEMBL1362545

SCHEMBL1362545

CCOC(=O)c1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC28A1 O00337 1/20 0.48
SLC28A2 O43868 1/20 0.48
SLC29A1 Q99808 1/20 0.48
SLC28A3 Q9HAS3 1/20 0.48
CDK1 P06493 1/20 0.44
P2RY2 P41231 1/20 0.43
PYGM P11217 3/20 0.41
UMPS P11172 1/20 0.39
SLC5A2 P31639 1/20 0.38
PNP P00491 1/20 0.38
TK2 O00142 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1362548 1.00 SLC28A1 (0.48) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL12143136 1.00 SLC28A1 (0.48) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL13455737 1.00 SLC28A1 (0.48) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL1362618 0.89 SLC28A1 (0.50) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL12143132 0.89 SLC28A1 (0.50) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL12143855 0.89 SLC28A1 (0.50) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL1362616 0.89 SLC28A1 (0.50) SLC28A1SLC28A2SLC29A1SLC28A3CDK1
SCHEMBL1361957 0.86 UMPS (0.58) P2RY2UMPS
SCHEMBL12143135 0.86 UMPS (0.58) P2RY2UMPS
SCHEMBL27744486 0.85 ENTPD2 (0.38) P2RY2UMPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931691-B1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIV HEALTH NETWORK (CA) 2013-08-21 EP claimed
US-8067391-B2 ODCase inhibitors for the treatment of malaria UNIVERSITY HEALTH NETWORK (CA) 2011-11-29 US claimed
US-20090221524-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIVERSITY HEALTH NETWORK (CA) 2009-09-03 US claimed
EP-1931691-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA University Health Network (CA) 2008-06-18 EP claimed
WO-2007038859-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIVERSITY HEALTH NETWORK (CA) 2007-04-12 WO claimed
EP-1931691-B1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIV HEALTH NETWORK (CA) 2013-08-21 EP disclosed
US-8067391-B2 ODCase inhibitors for the treatment of malaria UNIVERSITY HEALTH NETWORK (CA) 2011-11-29 US disclosed
US-20100056468-A1 Pyrimidine Derivatives As Anticancer Agents UNIVERSITY HEALTH NETWORK (CA) 2010-03-04 US disclosed
US-20090221524-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIVERSITY HEALTH NETWORK (CA) 2009-09-03 US disclosed
WO-2008083465-A1 PYRIMIDINE DERIVATIVES AS ANTICANCER AGENTS UNIVERSITY HEALTH NETWORK (CA) 2008-07-17 WO disclosed
EP-1931691-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA University Health Network (CA) 2008-06-18 EP disclosed
WO-2007038859-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UNIVERSITY HEALTH NETWORK (CA) 2007-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221524-A1 ODCASE INHIBITORS FOR THE TREATMENT OF MALARIA UMPS, UGDH, UPP1 SLC28A1 415/4885SLC28A2 455/4885SLC29A1 271/4885
US-20100056468-A1 Pyrimidine Derivatives As Anticancer Agents DPYD, TYMP, TYMS SLC28A1 165/4885SLC28A2 198/4885SLC29A1 58/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.