SCHEMBL13625503

SCHEMBL13625503

COCCNc1cc(CN(C(=O)[C@@H]2CCCNC2)C2CC2)c2ccccc2c1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.52
KCNH2 Q12809 5/20 0.47
CYP3A4 P08684 3/20 0.47
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13625505 0.85 REN (0.59) RENKCNH2CYP3A4
SCHEMBL13625586 0.84 REN (0.62) RENKCNH2CYP3A4
SCHEMBL13625504 0.79 REN (0.64) RENKCNH2CYP3A4
SCHEMBL13625497 0.78 REN (0.48) RENKCNH2CYP3A4SLC6A2SLC6A4
SCHEMBL12837185 0.78 REN (0.79) RENKCNH2CYP3A4
SCHEMBL1518210 0.78 REN (0.79) RENKCNH2CYP3A4
SCHEMBL1518212 0.78 REN (0.79) RENKCNH2CYP3A4
SCHEMBL12764077 0.78 REN (0.79) RENKCNH2CYP3A4
SCHEMBL1518206 0.78 REN (0.79) RENKCNH2CYP3A4
SCHEMBL13625565 0.73 REN (0.64) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009135299-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-11-12 WO disclosed