SCHEMBL13625587

SCHEMBL13625587

COCCCc1cc(CN(C(=O)[C@@H]2CCCNC2)C2CC2)c2ncccc2c1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
REN P00797 20/20 0.65
KCNH2 Q12809 10/20 0.65
CYP3A4 P08684 5/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13625591 0.88 REN (0.51) RENKCNH2CYP3A4
SCHEMBL13625586 0.87 REN (0.62) RENKCNH2CYP3A4
SCHEMBL13625505 0.83 REN (0.59) RENKCNH2CYP3A4
SCHEMBL13625565 0.82 REN (0.64) RENKCNH2CYP3A4
SCHEMBL13625584 0.81 REN (0.56) RENKCNH2CYP3A4
SCHEMBL13625727 0.81 REN (0.68) RENKCNH2CYP3A4
SCHEMBL13625716 0.81 REN (0.58) RENKCNH2CYP3A4
SCHEMBL13625728 0.81 REN (0.60) RENKCNH2CYP3A4
SCHEMBL13625717 0.81 REN (0.58) RENKCNH2CYP3A4
SCHEMBL1073071 0.80 REN (0.56) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009135299-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-11-12 WO disclosed