SCHEMBL13627227

SCHEMBL13627227

CNCc1cccc2ccc(-c3cccc(C(F)(F)F)c3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.47
CTSK P43235 4/20 0.47
KCNH2 Q12809 2/20 0.47
TRPV3 Q8NET8 1/20 0.45
KDM1A O60341 2/20 0.44
CNR2 P34972 2/20 0.41
CNR1 P21554 1/20 0.41
KMO O15229 1/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CG P48736 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
IDO1 P14902 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1032552 0.83 CTSS (0.47) CTSSCTSKKCNH2TRPV3KDM1A
SCHEMBL1034161 0.83 CTSS (0.47) CTSSCTSKKCNH2TRPV3KDM1A
SCHEMBL1034243 0.82 SCN9A (0.47) CTSSTRPV3KDM1AALDH1A1
SCHEMBL1034606 0.81 KDM1A (0.48) CTSSKDM1ACNR2
SCHEMBL13854087 0.81 CTSS (0.58) CTSSCTSKKDM1ACNR2KMO
SCHEMBL1035339 0.80 KIF11 (0.47) TRPV3KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL1033262 0.79 SCN9A (0.48) CTSSCTSKTRPV3KMOKDM4E
SCHEMBL1032856 0.76 KDM1A (0.50) CTSSKDM1AKMOPIK3CDPIK3CA
SCHEMBL28108403 0.75 NPSR1 (0.48) CTSSKDM1AKMOKDM4EALDH1A1
SCHEMBL27845626 0.73 CTSS (0.47) CTSSCTSKKDM1ACNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134973-A1 QUENOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed