SCHEMBL13627345

SCHEMBL13627345

COc1cc(NCc2ccccc2C(F)(F)F)cc2c1N(C)C[C@H]1CNC[C@@H]21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UTS2R Q9UKP6 4/20 0.40
EPHX2 P34913 2/20 0.38
CYP2D6 P10635 3/20 0.36
TSHR P16473 3/20 0.36
CYP2C19 P33261 3/20 0.36
MAPK1 P28482 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
HIF1A Q16665 1/20 0.36
ABL1 P00519 1/20 0.36
SRC P12931 1/20 0.36
GAA P10253 1/20 0.36
P2RX7 Q99572 1/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4488827 1.00 UTS2R (0.40) UTS2REPHX2CYP2D6TSHRCYP2C19
SCHEMBL13627340 0.88 GAA (0.38) UTS2REPHX2CYP3A4CYP2C9ABL1
SCHEMBL5955674 0.88 GAA (0.38) UTS2REPHX2CYP3A4CYP2C9ABL1
SCHEMBL4473034 0.88 GAA (0.38) UTS2REPHX2CYP3A4CYP2C9ABL1
SCHEMBL13627343 0.86 EGFR (0.36) CYP2C19CYP1A2CYP3A4GAAP2RX7
SCHEMBL4473434 0.86 EGFR (0.36) CYP2C19CYP1A2CYP3A4GAAP2RX7
SCHEMBL13627347 0.80 P2RX7 (0.38) UTS2REPHX2CYP2D6CYP1A2CYP3A4
SCHEMBL4480936 0.80 P2RX7 (0.38) UTS2REPHX2CYP2D6CYP1A2CYP3A4
SCHEMBL4477909 0.80 P2RX7 (0.38) UTS2REPHX2CYP2D6CYP1A2CYP3A4
SCHEMBL3130191 0.78 GAA (0.41) UTS2REPHX2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618980-B2 Pyrrolo(oxo)quinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-17 US disclosed