SCHEMBL13627408

SCHEMBL13627408

COc1ccc(-n2nc(C(=O)N3CC(N(C)C)C3(C)C)cc2-c2ccccn2)cn1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 8/20 0.35
MGLL Q99685 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
PIK3CD O00329 4/20 0.34
PIK3CA P42336 4/20 0.34
MALT1 Q9UDY8 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
PDK2 Q15119 1/20 0.33
SLC16A3 O15427 1/20 0.33
SLC16A1 P53985 1/20 0.33
RPA1 P27694 1/20 0.33
PIK3R2 O00459 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3R5 Q8WYR1 1/20 0.32
PIK3R3 Q92569 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2914121 0.89 RPA1 (0.45) MGLLMALT1RPA1
SCHEMBL2917841 0.84 MALT1 (0.44) NTRK1MGLLHCRTR1HCRTR2MALT1
SCHEMBL2920770 0.82 MALT1 (0.54) NTRK1MGLLMALT1
SCHEMBL5268929 0.80 MGLL (0.38) NTRK1MGLLHCRTR1HCRTR2PIK3CD
SCHEMBL2921813 0.80 NTRK1 (0.51) NTRK1MGLLPIK3CDPIK3CAMALT1
SCHEMBL2916328 0.79 BRD4 (0.41) NTRK1MGLLHCRTR1HCRTR2PIK3CD
SCHEMBL2919121 0.79 HCRTR1 (0.40) NTRK1MGLLHCRTR1HCRTR2PIK3CD
SCHEMBL2918250 0.79 RPA1 (0.52) NTRK1RPA1
SCHEMBL13637539 0.79 MALT1 (0.45) MGLLPIK3CDPIK3CAMALT1PIK3R2
SCHEMBL5531773 0.79 OXTR (0.39) NTRK1MALT1SLC16A3SLC16A1RPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622471-B2 Pyrazole derivatives having a pyridazine and pyridine functionality DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2009-11-24 US disclosed
US-7622471-B2 Pyrazole derivatives having a pyridazine and pyridine functionality DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2009-11-24 US disclosed