SCHEMBL13629395

SCHEMBL13629395

O=C1CCn2c1cc1ncccc12

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 1/20 0.34
PDE4A P27815 4/20 0.33
MET P08581 1/20 0.32
DAO P14920 2/20 0.32
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
THPO P40225 1/20 0.31
HIF1A Q16665 1/20 0.31
RAPGEF4 Q8WZA2 1/20 0.31
CDC7 O00311 1/20 0.31
CDK2 P24941 1/20 0.31
ATAD2 Q6PL18 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
BLM P54132 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30954503 0.78 PARP1 (0.44) CDC7
SCHEMBL27311284 0.78 PARP1 (0.44) CDC7
SCHEMBL18330320 0.74 PDE4A (0.52) PDE4A
SCHEMBL22490639 0.74 HRH3 (0.37) PDE4ACYP3A4
SCHEMBL30489158 0.74 PDE4A (0.52) PDE4A
SCHEMBL18527085 0.70 KDM4E (0.47) RPS6KA5LMNAMAPT
SCHEMBL1770250 0.70 NOTUM (0.35) RPS6KA5METDAOTSHRRAPGEF4
SCHEMBL569208 0.69 HPGD (0.42) RPS6KA5LMNA
SCHEMBL1253057 0.69 RXFP1 (0.35)
SCHEMBL21292094 0.68 PDE4A (0.49) PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618979-B2 Pyridopyrrolizine and pyridoindolizine derivatives MERCK FROSST CANADA LTD. (CA) 2009-11-17 US disclosed