SCHEMBL30954503

SCHEMBL30954503

O=C1NCCn2c1cc1ncccc12

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.44
RPS6KA3 P51812 8/20 0.44
MAPKAPK2 P49137 3/20 0.44
HRH3 Q9Y5N1 5/20 0.41
RPS6KA2 Q15349 5/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
CDC7 O00311 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27311284 1.00 PARP1 (0.44) PARP1RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL13629395 0.78 RPS6KA5 (0.34) CDC7
SCHEMBL27312316 0.77 RPS6KA3 (0.38) PARP1RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL1393632 0.76 RPS6KA3 (0.53) PARP1RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL30172384 0.76 RPS6KA3 (0.53) PARP1RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL22578499 0.76 PARP1 (0.53) PARP1RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL30954512 0.74 MAPKAPK2 (0.47) RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL30954513 0.74 MAPKAPK2 (0.47) RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL27311469 0.74 MAPKAPK2 (0.47) RPS6KA3MAPKAPK2HRH3RPS6KA2
SCHEMBL27312679 0.74 MAPKAPK2 (0.47) RPS6KA3MAPKAPK2HRH3RPS6KA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024118524-A1 AZAINDOLE COMPOUNDS AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS CEREVEL THERAPEUTICS, LLC (US) 2024-06-06 WO disclosed