SCHEMBL13629593

SCHEMBL13629593

COc1ccc(-n2ccnn2)cc1C=O

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.52
ALDH1A1 P00352 4/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KEAP1 Q14145 1/20 0.41
CYP19A1 P11511 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311297 0.80 KCNJ1 (0.54) NOTUMALDH1A1HPGDTSHR
SCHEMBL13629601 0.79 NOTUM (0.58) NOTUMKEAP1CYP19A1HCRTR1HCRTR2
SCHEMBL5193938 0.75 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL30412896 0.75 NOTUM (0.66) NOTUMKEAP1CYP19A1
SCHEMBL6540845 0.74 CYP11B1 (0.54) NOTUMALDH1A1CYP19A1POLB
SCHEMBL31402235 0.73 ALDH1A1 (0.40) NOTUMALDH1A1CYP1A2CYP2C9HPGD
SCHEMBL7120569 0.71 MAPT (0.50) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL4205532 0.70 ATM (0.45) NOTUMALDH1A1CYP1A2CYP2C9HPGD
SCHEMBL8530040 0.70 ALDH1A1 (0.40) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL31402350 0.70 FGFR1 (0.40) NOTUMALDH1A1CYP1A2CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed