SCHEMBL13629601

SCHEMBL13629601

COc1ccc(-n2ccnn2)cc1C

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 13/20 0.58
KEAP1 Q14145 1/20 0.45
CYP19A1 P11511 1/20 0.44
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
KMT2A Q03164 1/20 0.38
DBH P09172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15889924 0.81 NOTUM (0.63) NOTUMKEAP1CYP19A1
SCHEMBL30413228 0.81 NOTUM (0.63) NOTUMKEAP1CYP19A1
SCHEMBL30412896 0.79 NOTUM (0.66) NOTUMKEAP1CYP19A1
SCHEMBL13629593 0.79 NOTUM (0.52) NOTUMKEAP1CYP19A1HCRTR1HCRTR2
SCHEMBL16911508 0.77 NOTUM (0.46) NOTUMHCRTR1HCRTR2KMT2A
SCHEMBL16787394 0.77 NOTUM (0.58) NOTUMKEAP1CYP19A1
SCHEMBL4564455 0.77 NOTUM (0.58) NOTUMKEAP1CYP19A1
SCHEMBL16911330 0.75 HTT (0.44) KMT2ADBH
SCHEMBL20437909 0.74 NOTUM (0.58) NOTUMKEAP1CYP19A1
SCHEMBL28166936 0.74 NOTUM (0.67) NOTUMKEAP1CYP19A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed