SCHEMBL13629600

SCHEMBL13629600

CCOc1ccc(-n2nnnc2C(F)(F)F)cc1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
TACR1 P25103 10/20 0.44
NOTUM Q6P988 1/20 0.40
ALDH1A1 P00352 4/20 0.40
HSP90AA1 P07900 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
OXTR P30559 1/20 0.38
KCNN4 O15554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13629596 0.85 TACR1 (0.46) TACR1NOTUMALDH1A1HSP90AA1MAPT
SCHEMBL4203119 0.83 TACR1 (0.43) LMNATACR1
SCHEMBL13629602 0.82 TACR1 (0.46) TACR1NOTUMALDH1A1HSP90AA1MAPT
SCHEMBL4215358 0.80 MAPT (0.52) LMNANOTUMALDH1A1HSP90AA1MAPT
SCHEMBL4205359 0.79 ALDH1A1 (0.57) LMNATACR1NOTUMALDH1A1MAPT
SCHEMBL6541068 0.78 NOTUM (0.46) LMNATACR1NOTUMALDH1A1HSP90AA1
SCHEMBL4205786 0.77 MAPK1 (0.53) LMNAALDH1A1HPGDTSHRPOLB
SCHEMBL13630147 0.77 TACR1 (0.46) TACR1NOTUMALDH1A1HSP90AA1MAPT
SCHEMBL8517947 0.74 NOTUM (0.45) LMNATACR1NOTUMALDH1A1HSP90AA1
SCHEMBL8322001 0.74 TACR1 (0.38) TACR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed