SCHEMBL13630723

SCHEMBL13630723

NC(=O)Nc1[nH]c(-c2cccc(Oc3ccc(N)cc3)c2)cc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MITF O75030 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
GFER P55789 1/20 0.43
NLRP1 Q9C000 1/20 0.43
NOD2 Q9HC29 1/20 0.43
BRD4 O60885 4/20 0.42
CDC7 O00311 2/20 0.42
PARP10 Q53GL7 2/20 0.40
TNKS O95271 1/20 0.40
PARP15 Q460N3 1/20 0.40
PARP14 Q460N5 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200910 0.86 KDM4E (0.47) ALDH1A1MEN1KMT2AMAPTCDC7
SCHEMBL2198955 0.83 CDC7 (0.59) ALDH1A1SMN1; SMN2GAABRD4CDC7
SCHEMBL2199605 0.82 PARP1 (0.47) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL2201619 0.81 BRD4 (0.45) MEN1KMT2ABRD4CDC7IKBKB
SCHEMBL2197748 0.80 MAPT (0.48) ALDH1A1MEN1KMT2AGAAMAPT
SCHEMBL2200000 0.77 IKBKB (0.51) BRD4CDC7IKBKB
SCHEMBL2200529 0.77 CDC7 (0.40) SMN1; SMN2BRD4CDC7IKBKB
SCHEMBL2200146 0.77 BRD4 (0.62) BRD4CDC7IKBKB
SCHEMBL2196489 0.76 IKBKB (0.52) SMN1; SMN2MEN1KMT2ABRD4IKBKB
SCHEMBL2199810 0.76 CDC7 (0.56) BRD4CDC7IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2116530-A1 NOVEL PYRROLE DERIVATIVE HAVING UREIDE GROUP AND AMINOCARBONYL GROUP AS SUBSTITUENTS Santen Pharmaceutical Co., Ltd (JP) 2009-11-11 EP disclosed